ARL67156 trisodium hydrate is the trisodium hydrate salt form of ARL67156, a selective small-molecule inhibitor of ecto-ATPase enzymes including NTPDase1 (CD39), NTPDase3, and NPP1. Supplied as a white to off-white solid, it is intended for research use in studies of purinergic signaling, inflammation, and cardiovascular or respiratory disease models.
- Selective inhibitor of ecto-ATPase enzymes, including NTPDase1 (CD39), NTPDase3, and NPP1.
- Reported Kis values in the low micromolar range for primary targets.
- Demonstrated activity in cellular and tissue assays such as potentiation of neurogenic contractions and modulation of neurotransmitter release.
- High reported purity (99.94%), suitable for biochemical and cellular research.
- Supplied as a solid, white to off-white, available in small research quantities.